Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11996 |
MELK-8a hydrochloride
|
MELK | PI3K/Akt/mTOR signaling |
MELK-8a hydrochloride 是一种有效的母体胚胎亮氨酸拉链激酶抑制剂,IC50 为 2 nM。 | |||
T1759 |
OTSSP167
MELK inhibitor,OTS167 |
MELK | PI3K/Akt/mTOR signaling |
OTSSP167 (OTS167) 是一种高效的,ATP 竞争性的 MELK 抑制剂,其 IC50=0.41 nM。 | |||
T21559 |
OTSSP167 hydrochloride
OTSSP 167 盐酸盐 |
MELK | PI3K/Akt/mTOR signaling |
OTSSP167 hydrochloride 是一种高效的,ATP 竞争性的MELK 抑制剂,其 IC50=0.41 nM。 | |||
T11997 |
MELK-IN-1
Nintedanib Impurity L,MELK inhibitor 17,尼达尼布杂质L |
MELK | PI3K/Akt/mTOR signaling |
MELK-IN-1 (MELK inhibitor 17)是一种母体胚胎亮氨酸拉链激酶的有效抑制剂,IC50=3 nM,Ki=0.39 nM。 | |||
T24152 |
HTH-01-091
HTH-01091,HTH01-091,HTH 01-091,HTH 01091 |
Serine/threonin kinase; Pim; MELK; DYRK; CDK; RIP kinase | Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; JAK/STAT signaling; Metabolism; NF-κB; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors |
HTH-01-091 是一种强效且选择性的 maternal embryonic leucine zipper kinase (MELK) 抑制剂(IC50 :10.5 nM)。HTH-01-091 对PIM1/2/3、RIPK2、DYRK3、smMLCK 和 CLK2有抑制作用。HTH-01-091 可用于研究乳腺癌。 | |||
T70578 | BX-795 hydrochloride | ||
BX-795 hydrochloride is a TBK1 and IKKε inhibitor. BX-795 is a potential maternal embryonic leucine zipper kinase inhibitor. | |||
T73867 | HTH-01-091 TFA | ||
HTH-01-091 TFA 是一种强效且选择性的maternal embryonic leucine zipper kinase (MELK)抑制剂,其IC50为 10.5 nM。HTH-01-091 TFA 还能抑制PIM1/2/3、RIPK2、DYRK3、smMLCK 和CLK2。HTH-01-091 TFA 可用于乳腺癌研究。 |